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Application of bioisosteres to modulate molecular properties in medicinal chemistry
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The development of chemo- and regioselective reactions of boron systems
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Targeted protein degradation as a new approach to drug discovery
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Development towards prospective modelling of in vivo rabbit QTc prolongation
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Pharmacological characterisation of the 5-HT receptors present on mouse and human hepatic stellate cells and their role in liver fibrosis
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Single electron transfer in organic synthesis targeted towards sustainable manufacture
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Mechanistic pharmacokinetic / pharmacodynamic modelling of acute inflammatory challenge models
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Studies and improvement of molecular docking methods in rigid and flexible receptors
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Development of the C-methyltransferases NovO and CouO for biocatalytic Friedel-Crafts alkylation
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