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Studies towards the synthesis and labelling of bioactive peptides
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The design and synthesis of probe molecules to validate the inhibition of epigenetic mechanisms for phenotypic responses
2 di 20
Development of chemical probes for non-BET bromodomains
3 di 20
Novel biocatalytic strategies for the synthesis of N-functionalised amino acids
4 di 20
New methods for the synthesis of pharmaceutical azacycles
5 di 20
Development of photoaffinity labelling technologies for small molecule drug discovery - a case study targeting bromodomains
6 di 20
Application of electrochemical based sensors in support of toxicokinetic and pharmacokinetics
7 di 20
The development of small molecules for treatment of idiopathic pulmonary fibrosis (IPF)
8 di 20
The design and synthesis of small molecule bromodomain inhibitors
9 di 20
The design and synthesis of targeted BET inhibitors
10 di 20
Novel C-C bond formation strategies for access to secondary and tertiary amides enabled by new synthetic technologies
11 di 20
Novel approaches targeting phosphoinositide 3-kinase delta
12 di 20
Synthesis and optimisation of novel molecules to probe epigenetic mechanisms with applications in the treatment of inflammatory disorders
13 di 20
Development of lysine acylating small molecules for covalent kinase inhibition
14 di 20
Investigating streptomyces clavuligerus linear replicons for improved clavulanic acid production
15 di 20
Design and synthesis of dimethylisoxazole quinolines as BET inhibitors
16 di 20
The development and evaluation of a method for the quantitative determination of a monoclonal antibody using capillary electrophoresis-high resolution mass spectrometry
17 di 20
Pharmacological characterisation of the 5-HT receptors present on mouse and human hepatic stellate cells and their role in liver fibrosis
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The application of flow chemistry to the synthesis of pharmaceutically privileged heterocycles
19 di 20
Chan-Lam animation studies : solving the chemotype reactivity issue
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