Development of photoaffinity labelling technologies for small molecule drug discovery - a case study targeting bromodomains

New methods for the synthesis of pharmaceutical azacycles

The design and synthesis of chemical probes for non-BET bromodomains

Development of chemical probes for non-BET bromodomains

The design and synthesis of small molecule bromodomain inhibitors

Sustainable cross-couplings for pharmaceutical scale-up using aryldiazonium salts