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Development and understanding of rhodium-catalysed conjugate arylation for process chemistry applications
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Synthesis and biological evaluation of novel small molecule bromodomain inhibitors
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Synthesis of non-natural base-pairs : towards site-specific functionalisation of nucleic acids
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Development of small molecule splice-switchers as inducers of apoptosis
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New chemical approaches for the development of targeted protein degradation
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Chemoselective C-H functionalisation of aliphatic azacycles : utilisation of electrophilic iodine as a mild oxidant
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Development of novel inhibitors of carbohydrate-processing targets involved in Mycobacterium tuberculosis cell wall biosynthesis
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Development of the C-methyltransferases NovO and CouO for biocatalytic Friedel-Crafts alkylation
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