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Jamieson, Craig
删除限定条件 贡献者: Jamieson, Craig
部门,学校或学院
Department of Pure and Applied Chemistry
删除限定条件 部门,学校或学院: Department of Pure and Applied Chemistry
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Synthesis and evaluation of novel small molecule inhibitors of the androgen receptor amino-terminal domain for the treatment of castration-resistant prostate cancer
创造者:
Riley, Christopher
日期:
2021
Department, School or Faculty:
Department of Pure and Applied Chemistry
The design, synthesis and optimisation of calcium release-activated calcium (CRAC) channel inhibitors and mitochondrial permeability transition pore (mPTP) modulators, using phenotypic screening
创造者:
Lacroix, Yannick
日期:
2015
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
The design and synthesis of αvβ6 antagonists and PI3K inhibitors as small molecule therapies for respiratory diseases
创造者:
Tame, Christopher J.
日期:
2014
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Studies towards the synthesis and labelling of bioactive peptides
创造者:
Stewart, Sam
日期:
2016
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Investigation and application of 3-Oxabicyclo[4.1.0]heptane as a mechanistic target of rapamycin (mTOR) kinase hinge binding fragment
创造者:
Summers, Declan M.
日期:
2019
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Structure-guided discovery of a novel steroid-derived family of autotaxin inhibitors based on endogenous allosteric modulators
创造者:
Clark, Jennifer M.
日期:
2020 and 2021
Department, School or Faculty:
Department of Pure and Applied Chemistry
Structure-guided approaches to the design of novel autotaxin inhibitors
创造者:
Potjewyd, Frances
日期:
2016
Funder:
Engineering and Physical Sciences Research Council
and
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
The synthesis and optimisation of toll-like receptor agonists as potential immunomodulatory agents
创造者:
Tape, Daniel Terence
日期:
2016
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Investigation of LPA₁ receptor antagonism / ATX inhibition by a scaffold hopping aproach and SAR analysis
创造者:
Castagna, Diana
日期:
2016
Department, School or Faculty:
Department of Pure and Applied Chemistry
The development of natural products as phytotoxic leads for herbicide discovery
创造者:
Littleson, Mairi M.
日期:
2017
Department, School or Faculty:
Department of Pure and Applied Chemistry
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28
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Doctoral thesis
28
创造者
Campbell, Peter
1
Castagna, Diana
1
Clark, Jennifer M.
1
Duffy, Emma
1
Green, Luke
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贡献者
Jamieson, Craig
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28
GlaxoSmithKline
15
Watson, Allan
6
Engineering and Physical Sciences Research Council
2
Hirst, David
2
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出资者
GlaxoSmithKline
15
Engineering and Physical Sciences Research Council
2
Carnegie Trust for the Universities of Scotland
1
Gyros Protein Technologies
1
部门,学校或学院
Department of Pure and Applied Chemistry
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28
日期
2016
6
2018
5
2020
4
2021
4
2022
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