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Jamieson, Craig
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Synthesis and evaluation of novel small molecule inhibitors of the androgen receptor amino-terminal domain for the treatment of castration-resistant prostate cancer
Creador:
Riley, Christopher
Fecha:
2021
Department, School or Faculty:
Department of Pure and Applied Chemistry
The design, synthesis and optimisation of calcium release-activated calcium (CRAC) channel inhibitors and mitochondrial permeability transition pore (mPTP) modulators, using phenotypic screening
Creador:
Lacroix, Yannick
Fecha:
2015
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
The design and synthesis of αvβ6 antagonists and PI3K inhibitors as small molecule therapies for respiratory diseases
Creador:
Tame, Christopher J.
Fecha:
2014
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Studies towards the synthesis and labelling of bioactive peptides
Creador:
Stewart, Sam
Fecha:
2016
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Investigation and application of 3-Oxabicyclo[4.1.0]heptane as a mechanistic target of rapamycin (mTOR) kinase hinge binding fragment
Creador:
Summers, Declan M.
Fecha:
2019
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Structure-guided discovery of a novel steroid-derived family of autotaxin inhibitors based on endogenous allosteric modulators
Creador:
Clark, Jennifer M.
Fecha:
2020 and 2021
Department, School or Faculty:
Department of Pure and Applied Chemistry
Structure-guided approaches to the design of novel autotaxin inhibitors
Creador:
Potjewyd, Frances
Fecha:
2016
Funder:
Engineering and Physical Sciences Research Council
and
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
The synthesis and optimisation of toll-like receptor agonists as potential immunomodulatory agents
Creador:
Tape, Daniel Terence
Fecha:
2016
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Investigation of LPA₁ receptor antagonism / ATX inhibition by a scaffold hopping aproach and SAR analysis
Creador:
Castagna, Diana
Fecha:
2016
Department, School or Faculty:
Department of Pure and Applied Chemistry
The development of natural products as phytotoxic leads for herbicide discovery
Creador:
Littleson, Mairi M.
Fecha:
2017
Department, School or Faculty:
Department of Pure and Applied Chemistry
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Jamieson, Craig
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GlaxoSmithKline
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Watson, Allan
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Engineering and Physical Sciences Research Council
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Carnegie Trust for the Universities of Scotland
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Gyros Protein Technologies
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Department of Pure and Applied Chemistry
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Strathclyde Institute of Pharmacy and Biomedical Sciences
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