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Jamieson, Craig
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Risultati della ricerca
Exploiting DNA-encoded library : technology for the discovery of novel antibody recruiting molecules against LOX-1
Creatore:
Macfarlane, Katherine F.
Data:
2022
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Development of new synthetic approaches in solid-phase peptide synthesis
Creatore:
Mowat, Jenna Marie
Data:
2023 and 2024
Funder:
Gyros Protein Technologies
Department, School or Faculty:
Department of Pure and Applied Chemistry
Computer-aided drug design of bicyclic-derived BRD4 inhibitors
Creatore:
Little, Gemma
Data:
2023
Funder:
Engineering and Physical Sciences Research Council
Department, School or Faculty:
Department of Pure and Applied Chemistry
Synthetic approaches to heterocyclic systems of pharmaceutical relevance
Creatore:
Green, Luke
Data:
2021
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Homogeneous hydrogenation and photochemistry as tools in pharmaceutical process development
Creatore:
Shaalan, Youssef
Data:
2021
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Application of bioisosteres to modulate molecular properties in medicinal chemistry
Creatore:
Measom, Nicholas
Data:
2017
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
The use of contemporary chemoproteomic techniques in antimalarial target identification
Creatore:
Tucker, Jessie S.
Data:
2020
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Application of computer vision in industrially important reactions
Creatore:
Yan, Chunhui
Data:
2022
Department, School or Faculty:
Department of Pure and Applied Chemistry
Development of new chemical tools as crop protecting agents
Creatore:
Hamer, Meghan M.
Data:
2022
Department, School or Faculty:
Department of Pure and Applied Chemistry
Novel approaches targeting phosphoinositide 3-kinase delta
Creatore:
Spencer, Jonathan Andrew
Data:
2018
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Synthesis and evaluation of novel small molecule inhibitors of the androgen receptor amino-terminal domain for the treatment of castration-resistant prostate cancer
Creatore:
Riley, Christopher
Data:
2021
Department, School or Faculty:
Department of Pure and Applied Chemistry
The design, synthesis and optimisation of calcium release-activated calcium (CRAC) channel inhibitors and mitochondrial permeability transition pore (mPTP) modulators, using phenotypic screening
Creatore:
Lacroix, Yannick
Data:
2015
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
The design and synthesis of αvβ6 antagonists and PI3K inhibitors as small molecule therapies for respiratory diseases
Creatore:
Tame, Christopher J.
Data:
2014
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Studies towards the synthesis and labelling of bioactive peptides
Creatore:
Stewart, Sam
Data:
2016
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Investigation and application of 3-Oxabicyclo[4.1.0]heptane as a mechanistic target of rapamycin (mTOR) kinase hinge binding fragment
Creatore:
Summers, Declan M.
Data:
2019
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Structure-guided discovery of a novel steroid-derived family of autotaxin inhibitors based on endogenous allosteric modulators
Creatore:
Clark, Jennifer M.
Data:
2020 and 2021
Department, School or Faculty:
Department of Pure and Applied Chemistry
Structure-guided approaches to the design of novel autotaxin inhibitors
Creatore:
Potjewyd, Frances
Data:
2016
Funder:
Engineering and Physical Sciences Research Council
and
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
The synthesis and optimisation of toll-like receptor agonists as potential immunomodulatory agents
Creatore:
Tape, Daniel Terence
Data:
2016
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Investigation of LPA₁ receptor antagonism / ATX inhibition by a scaffold hopping aproach and SAR analysis
Creatore:
Castagna, Diana
Data:
2016
Department, School or Faculty:
Department of Pure and Applied Chemistry
The development of natural products as phytotoxic leads for herbicide discovery
Creatore:
Littleson, Mairi M.
Data:
2017
Department, School or Faculty:
Department of Pure and Applied Chemistry
Development of novel allosteric regulators of proteinase-activated receptors
Creatore:
Sloan, Graeme McDermott
Data:
2019
Department, School or Faculty:
Strathclyde Institute of Pharmacy and Biomedical Sciences
Investigations into the generation and pleiotropic reactivity modes of the nitrile imine 1,3-dipole
Creatore:
Livingstone, Keith
Data:
2020
Department, School or Faculty:
Department of Pure and Applied Chemistry
Approaches to lead generation for idiopathic pulmonary fibrosis targets
Creatore:
Duffy, Emma
Data:
2016
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
New methods for the construction of selectively difluorinated carbocycles
Creatore:
McCarter, Adam William
Data:
2018
Funder:
GlaxoSmithKline
and
Carnegie Trust for the Universities of Scotland
Department, School or Faculty:
Department of Pure and Applied Chemistry
The development of novel organocatalytic and transition-metal catalysed methodologies for amide bond formation
Creatore:
McPherson, Christopher
Data:
2018
Department, School or Faculty:
Department of Pure and Applied Chemistry
The design and synthesis of molecular tools for probing biological function
Creatore:
Milne, Kirsty
Data:
2020 and 2019
Department, School or Faculty:
Department of Pure and Applied Chemistry
Expedient access to C-aryl linked saturated heterocyclic motifs
Creatore:
Campbell, Peter
Data:
2018
Department, School or Faculty:
Department of Pure and Applied Chemistry
The development of small molecule inhibitors for fibrosis drug discovery
Creatore:
Miller, Lisa Margaret
Data:
2016
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Evaluating the application and limitations of bio-based solvents within organic synthesis
Creatore:
Wilson, Kirsty Leanne
Data:
2018
Department, School or Faculty:
Department of Pure and Applied Chemistry
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Thesis
29
Tipo di risorsa
Doctoral thesis
29
Creatore
Campbell, Peter
1
Castagna, Diana
1
Clark, Jennifer M.
1
Duffy, Emma
1
Green, Luke
1
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Collaboratore
Jamieson, Craig
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29
GlaxoSmithKline
15
Watson, Allan
6
Engineering and Physical Sciences Research Council
2
Hirst, David
2
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Funder
GlaxoSmithKline
15
Engineering and Physical Sciences Research Council
2
Carnegie Trust for the Universities of Scotland
1
Gyros Protein Technologies
1
Dipartimento, Scuola o Facoltà
Department of Pure and Applied Chemistry
28
Strathclyde Institute of Pharmacy and Biomedical Sciences
1
Data
2016
6
2018
5
2020
4
2021
4
2019
3
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