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Novel heterocyclic ligands for the lipid kinase PI4KIIIβ : a chemical biology approach
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Development of photoaffinity labelling technologies for small molecule drug discovery - a case study targeting bromodomains
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New methods for the synthesis of pharmaceutical azacycles
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The design and synthesis of chemical probes for non-BET bromodomains
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Preclinical development of a treatment for systemic lupus erythematosus
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Development of chemical probes for non-BET bromodomains
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The design and synthesis of small molecule bromodomain inhibitors
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Sustainable cross-couplings for pharmaceutical scale-up using aryldiazonium salts
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