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Application of bioisosteres to modulate molecular properties in medicinal chemistry
1 de 9
The development of chemo- and regioselective reactions of boron systems
2 de 9
Targeted protein degradation as a new approach to drug discovery
3 de 9
Development towards prospective modelling of in vivo rabbit QTc prolongation
4 de 9
Pharmacological characterisation of the 5-HT receptors present on mouse and human hepatic stellate cells and their role in liver fibrosis
5 de 9
Single electron transfer in organic synthesis targeted towards sustainable manufacture
6 de 9
Mechanistic pharmacokinetic / pharmacodynamic modelling of acute inflammatory challenge models
7 de 9
Studies and improvement of molecular docking methods in rigid and flexible receptors
8 de 9
Development of the C-methyltransferases NovO and CouO for biocatalytic Friedel-Crafts alkylation
9 de 9