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Development and understanding of rhodium-catalysed conjugate arylation for process chemistry applications
1 de 10
Synthesis and biological evaluation of novel small molecule bromodomain inhibitors
2 de 10
Understanding the hepatic disposition of statins to improve predictions of safety and efficacy
3 de 10
The design and synthesis of chemical probes for non-BET bromodomains
4 de 10
New dose estimation methods and their application in early drug discovery using intravenous, oral and inhaled routes of administration for new chemical entities
5 de 10
New chemical approaches for the development of targeted protein degradation
6 de 10
Investigation and application of 3-Oxabicyclo[4.1.0]heptane as a mechanistic target of rapamycin (mTOR) kinase hinge binding fragment
7 de 10
The application of flow chemistry to the synthesis of pharmaceutically privileged heterocycles
8 de 10
Understanding reaction mechanisms and structure/reactivity relationships in the electrophilic fluorination of enol esters
9 de 10
Automated, quantitative process analysis by NMR
10 de 10