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The design and synthesis of probe molecules to validate the inhibition of epigenetic mechanisms for phenotypic responses
Schöpfer:
Hayhow, Thomas G.
Datum:
2014
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Development towards prospective modelling of in vivo rabbit QTc prolongation
Schöpfer:
Lewis, Gareth John
Datum:
2017
Funder:
GlaxoSmithKline
Department, School or Faculty:
Strathclyde Institute of Pharmacy and Biomedical Sciences
Chan-Lam animation studies : solving the chemotype reactivity issue
Schöpfer:
Vantourout, Julien
Datum:
2018
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Chemoselective C-H functionalisation of aliphatic azacycles : utilisation of electrophilic iodine as a mild oxidant
Schöpfer:
Griffiths, Robert Joseph
Datum:
2018
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Investigation and application of 3-Oxabicyclo[4.1.0]heptane as a mechanistic target of rapamycin (mTOR) kinase hinge binding fragment
Schöpfer:
Summers, Declan M.
Datum:
2019
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
The application of flow chemistry to the synthesis of pharmaceutically privileged heterocycles
Schöpfer:
Baker, Blake Jamie Mark
Datum:
2019
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Iron-catalysed cross-couplings of secondary alkyl Grignard reagents
Schöpfer:
Sanderson, James
Datum:
2018
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Computational modelling of enzyme activity to speed up biocatalyst redesign
Schöpfer:
Dréanic, Marie-Pierre
Datum:
2018
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Increasing the saturation of BET inhibitors
Schöpfer:
Dixon, Joseph Edward
Datum:
2018
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
Understanding reaction mechanisms and structure/reactivity relationships in the electrophilic fluorination of enol esters
Schöpfer:
Wood, Susanna Helen
Datum:
2019
Funder:
GlaxoSmithKline
Department, School or Faculty:
Department of Pure and Applied Chemistry
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Jamieson, Craig
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Biotechnology and Biological Sciences Research Council
1
Carnegie Trust for the Universities of Scotland
1
EPSRC Centre for Doctoral Training in Technology Enhanced Chemical Synthesis
1
Engineering and Physical Sciences Research Council
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Department of Pure and Applied Chemistry
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Strathclyde Institute of Pharmacy and Biomedical Sciences
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WestCHEM
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