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Development of lysine acylating small molecules for covalent kinase inhibition
1 de 10
Novel heterocyclic ligands for the lipid kinase PI4KIIIβ : a chemical biology approach
2 de 10
A medicinal chemistry approach towards brodomain epigenetic modulators
3 de 10
Synthesis and optimisation of novel molecules to probe epigenetic mechanisms with applications in the treatment of inflammatory disorders
4 de 10
The development and evaluation of a method for the quantitative determination of a monoclonal antibody using capillary electrophoresis-high resolution mass spectrometry
5 de 10
The use of structure-based drug design to optimise protein-ligand interactions
6 de 10
The design, synthesis and optimisation of αvβ6 antagonists as potential idiopathic pulmonary fibrosis agents
7 de 10
Electrochemically enabled synthesis of substituted isoxazolines
8 de 10
αV integrin antagonists for the treatment of idiopathic pulmonary fibrosis
9 de 10
Application of electrochemical based sensors in support of toxicokinetic and pharmacokinetics
10 de 10