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The design and synthesis of targeted BET inhibitors
1 de 10
Novel C-C bond formation strategies for access to secondary and tertiary amides enabled by new synthetic technologies
2 de 10
Novel approaches targeting phosphoinositide 3-kinase delta
3 de 10
Synthesis of non-natural base-pairs : towards site-specific functionalisation of nucleic acids
4 de 10
Preclinical development of a treatment for systemic lupus erythematosus
5 de 10
Development of small molecule splice-switchers as inducers of apoptosis
6 de 10
Pharmacological characterisation of small molecule RGD-mimetics targeting αvβ6-mediated activation of TGFβ in idiopathic pulmonary fibrosis
7 de 10
The design, synthesis and optimisation of calcium release-activated calcium (CRAC) channel inhibitors and mitochondrial permeability transition pore (mPTP) modulators, using phenotypic screening
8 de 10
The design and synthesis of novel epigenetic modulators
9 de 10
Development of chemical probes for non-BET bromodomains
10 de 10