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The design and synthesis of αvβ6 antagonists and PI3K inhibitors as small molecule therapies for respiratory diseases
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Investigation of LPA₁ receptor antagonism / ATX inhibition by a scaffold hopping aproach and SAR analysis
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Evaluating the application and limitations of bio-based solvents within organic synthesis
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Computer-aided drug design of bicyclic-derived BRD4 inhibitors
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Novel approaches targeting phosphoinositide 3-kinase delta
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Development of new chemical tools as crop protecting agents
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Studies towards the synthesis and labelling of bioactive peptides
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Application of bioisosteres to modulate molecular properties in medicinal chemistry
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The use of contemporary chemoproteomic techniques in antimalarial target identification
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Synthesis and evaluation of novel small molecule inhibitors of the androgen receptor amino-terminal domain for the treatment of castration-resistant prostate cancer
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